Upadacitinib (Rinvoq): appropriate for treating inflammatory disorders such as:
Rheumatoid arthritis (adults)
Psoriatic arthritis (greater than two years of age)
Ankylosing spondylitis (adults)
A & B
B & C
A & C
A, B & C
Upadacitinib (Rinvoq): appropriate for treating inflammatory disorders such as:
Non-radiographic axial spondyloarthritis (adults)
Atopic dermatitis (greater than 12 years of age)
Ulcerative colitis (adults)
Crohn's disease (adults)
All of the above disorders may be treated with upadacitinib (Rinvoq).
Upadacitinib (Rinvoq): Not a first-choice treatment for inflammatory disorders; typically employed if other drugs such as adalimumab (Humira) administration
did not result in adequate responses.
True
False
JAK inhibitors
administration may elevate risk of certain serious adverse reactions including blood clots.
True
False
Upadacitinib (Rinvoq):
Second-line agent for treating moderate to severe rheumatoid arthritis in patients with inadequate response (or intolerant) to methotrexate, the first-line drug.
Classified as
a selective Janus kinase (JAK) inhibitor that targets the JAK1 enzyme.
Chrouos G Ch 39
Adrenocorticosteroids & Adrenocortical Antagonists in
Katzung's Basic & Clinical Pharmacology (Vanderah TW, ed)
16e McGraw Hill 2023
Brezinski E Klickstein L Armstrong A Ch 46 Pharmacology of
Immunosuppression in Principles of Pharmacology: The
Pathophysiologic Basis of Drug Therapy. (Golan DE Armstrong
EJ Armstrong AW, eds) 4e 2017
Ritter JM Flower R
Henderson G Loke YK MacEwan D Robinson E Fullerton J Ch 25
Anti-inflammatory and Immunosuppressant Drugs Rang & Dale's
Pharmacology 10e Elsevier 2024.
Burchum J Rosenthal L
Lehne's Pharmacology for Nursing Care Ch 72
Immunosuppressants Elsevier 2022.
Burchum J Rosenthal L
Lehne's Pharmacology for Nursing Care Ch 75 Glucocorticoids
in Nonendrocrine Disorders Elsevier 2022.
Burchum J Rosenthal L
Lehne's Pharmacology for Nursing Care Ch 76 Drug Therapy for
Rheumatoid Arthritis Elsevier 2022.
Bass A Rogatsky Ch 32
Immunomodulatory Drugs in Goldman-Cecil Medicine (Goldman L
Schafer, eds) Elsevier 26e 2020
Leiva M Takemoto Ch
238 Immunosuppressants in Lippincott Illustrated Reviews:
Pharmacology 8e ((Walen et al, eds) Wolters Kluwer 2023.
Hall J Hall M Ch 78
Adrenocortical Hormones Guyton and Hall Textbook of Medical
Physiology 14e Elsevier 2021.
Waller DG Sampson A
Hitchings Ch 38 The Immune Response and Immunosuppressant
Drugs Medical Pharmacology & Therapeutics 6e Elsevier
2022
Waller DG Sampson A
Hitchings Ch 30 Rheumotoid Arthritis, Other Inflammatory
Arthrides and Osteoarthritis Medical Pharmacology &
Therapeutics 6e Elsevier 2022